ALX550400M005
ENZOALX550400M005EA
192
EUR
InStock
ENZOALX550400M005
Dimethyl-W84 dibromide ≥98% (par HPLC)
Dimethyl-W84 dibromide
M2 receptor modulator.
Very potent allosteric modulator of muscarinic receptors, selective for M2-receptors.
Retards the dissociation of the antagonist N-methylscopolamine. Affinity for the free receptor is about 10-fold higher than with W84. pKA=7.08, p(αKA)=6.75, pEC₅₀,diss=6.77.
Soluble in DMSO, water or aqueous buffer.