ENZOALX380008M005EA
115.5
EUR
InStock
ENZOALX380008M005
ENZOALX380008M001
ENZOALX380008M025
Tacrolimus ≥98%, poudre cristalline
Tacrolimus
Immunosuppressant.
Immunosuppressant that blocks T cell proliferation in vitro by inhibiting the generation of several lymphokines, especially IL-2. Shown to inhibit the activity of FK506 binding protein and to inhibit the Ca²⁺-dependent phosphatase and protein phosphatase 2B (PP2B; calcineurin). Activates NF-κB through phosphorylation and degradation of IκBα.
Soluble in DMSO, 100% ethanol, methanol, ethyl acetate or acetone; insoluble in water.